Sl.No Name Structure CAS API
1. (1R,2R)-1-(tert-Butoxycarbo- nyl amino)-2-(difluoromethyl) cyclopropane carboxylic acid 1152134-45-6 Glecaprevir
(Mavyret)
2. 1-Methylcyclopropane sulfonamide 669008-26-8 Glecaprevir
(Mavyret)
3. (3S,5S,6R)-3-amino-6-methyl-5-phenyl-1-(2,2,2-trifluoroethyl)piperidin-2-one 1375794-69-6 Ubrogepant
(Ubrelvy)
4. (5S,6S,9R)-5-amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-ol 1373116-05-2 Rimegepant
(Nurtec ODT)
5. tert-Butyl-(1R, 2S, 5S)-2-amino-5-(dimethylcarbamoyl) cyclohexyl carbamate 365998-36-3 Edoxaban
6. 2-((6-chloro-3-methyl-2,4-dioxo3,4-dihydropyrimidin-1(2H)-yl)methyl)benzonitrile 865758-96-9 Commercial Alogliptin
7. 4-(Pyrrolidino Sulfonyl Methyl) Nitrobenzene 340041-91-0 Commercial Alomotriptan
8. 4-(Pyrrolidino Sulfonyl Methyl) Benzeneamine 334981-10-1 Commercial Alomotriptan
9. 4-Fluoro-3-nitrobenzonitrile 1009-35-4 Lab Scale Alectinib
10. 4-Morpholinopiperidine 53617-35-9 Lab Scale Alectinib
11. (2S)-1-[[(2-Amino-1,1-dimethyl ethyl)amino]acetyl]-2-pyrrolidinecarbonitrile 794460-89-2 Lab Scale Anagliptin
12. 2-methylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid 739364-95-5 Lab Scale Anagliptin
13. 2-Methyl-1,2-propanediamine 811-93-8 Lab Scale Anagliptin
14. 2-Formyl-3-oxo-propionic Acid Ethyl Ester 80370-42-9 Lab Scale Anagliptin
15. 3-Methyl-1H-pyrazol-5-amine 31230-17-8 Lab Scale Anagliptin
16. tert-Butyl (2-amino-2-methylpropyl)carbamate 95034-05-2 Lab Scale Anagliptin
17. 7-hydroxy-3,4-dihydroquinolin-2(1H)-one 22246-18-0 Commercial Aripiprazole
18. 1-(2,3-dichloro phenyl) piperazine hydrochloride 119532-26-2 Commercial Aripiprazole
19. 2,3-dihydro-N-phenyl-1H-inden-2-amine hydrochloride 33237-73-9 Lab scale Aprindine
20. (R)-4-Propylpyrrolidin-2-one 930123-37-8 Lab Scale Brivaracetam
21. (R)-4-propyl-dihydro-furan-2-one 63095-51-2 Lab Scale Brivaracetam
22. 3-(4-Chloro phenyl)glutaric acid 35271-74-0 Commercial Baclofen
23. 3-(4-chlorophenyl)glutaric acid monoamide 1141-23-1 Commercial Baclofen
24. 2-Bromo-5-Hydroxy Benzaldehyde 2973-80-0 Lab Scale Crisaborole
25. 4-(4-bromo-3-formylphenoxy)benzonitrile 906673-54-9 Lab Scale Crisaborole
26. Methyl 3-amino-2-fluorobenzoate 1195768-18-3 Lab Scale Dabrafenib
27. 1H-imidazole-4-carboxylic acid 1072-84-0 Commercial Dexmedetomidine
28. (2,3-dimethyl phenyl) magnesium bromide 134640-85-0 Commercial Dexmedetomidine
29. 4-(1-(2,3-dimethyl phenyl) vinyl)-1H-imidazole hydrochloride Lab Scale Dexmedetomidine
30. 3-[(3-Amino-4-methylamino-benzoyl)-pyridin-2-yl-amino]-propionic acid ethyl ester 212322-56-0 Pilot Scale Dabigitran
31. 3-(Pyridin-2-ylamino)-propionic acid ethyl ester 103041-38-9 Pilot Scale Dabigitran
32. (4-Cyano-phenylamino)-acetic acid 42288-26-6 Pilot Scale Dabigitran
33. 4-N-Methylamino-3-nitro benzoic acid 41263-74-5 Pilot Scale Dabigitran
34. (2-chloro-5-iodophenyl)(4-ethoxyphenyl)methanone 1103738-26-6 Pilot Scale Dapagliflozin
35. 1-(2-chloro-5-iodobenzyl)-4-ethoxybenzene 1103738-29-9 Pilot Scale Dapagliflozin
36. 4-Amino-2-chloro-6,7-dimethoxyquinazoline 23680-84-4 Commercial Doxazosin
37. (2-Chloro-5-iodophenyl)(4-fluorophenyl)methanone 915095-86-2 Pilot Scale Empagliflozin
38. (S)-(2-Chloro-5-iodophenyl) (4-(tetrahydrofuran-3-yloxy) phenyl)methanone 915095-87-3 Pilot Scale Empagliflozin
39. (3S)-3-(4-(2-chloro-5-iodobenzyl)phenoxy)tetrahydrofuran 915095-94-2 Pilot Scale Empagliflozin
40. 4(2-cyanopropan-2-ylamino)2-fluoro-N-methylbenzamide 915087-32-0 Lab Scale Enzalutamide
41. 4-isothiocyanato-2-(trifluoromethyl)benzonitrile 143782-23-4 Lab Scale Enzalutamide
42. 5-Bromo-3-(((R)-1-methyl pyrrolidine-2-yl) methyl)-1H-indole 143322-57-0 Commercial Eletriptan
43. Phenyl vinyl sulfone 5535-48-8 Commercial Eletriptan
44. 1-(2,3-dichloro-4-hydroxyphenyl)butan-1-one 2350-46-1 Commercial Ethacrynic Acid
45. (6RS)-6-Methylamino-6,7,8,9-tetrahydro-5H-carbazole-3-carbonitrile 147009-33-4 Lab Scale Frovatriptan
46. (6R)-6-Methylamino-6,7,8,9-tetrahydro-5H-carbazole-3-carbonitrile 247939-84-0 Lab Scale Frovatriptan
47. 3,3-Dimethyl-1,5-dioxa-spiro[5.5]undec-9-yl)-methyl-amine. Hydrochloride 158747-10-5 Lab Scale Frovatriptan
48. (1-(3-Trifluoro Methyl) Phenyl Piperazine 15532-75-9 Lab Scale Flibanserin
49. (1-(3-Trifluoro Methyl) Phenyl Piperazine 15532-75-9 Lab Scale Flibanserin
50. 1-(2-Chloro-ethyl)-1,3-dihydro-benzimidazol-2-one 52548-84-2 Lab Scale Flibanserin
51. 3-Cyano-4-isobutoxybenzamide 161718-85-0 Commercial Fabuxostat
52. 2-(2-butyl-4-hydroxy-6-methylpyrimidin-5-yl)-N,N-dimethylacetamide 1315478-13-7 Lab Scale Fimasatran
53. 4-Bromo-2-fluorobiphenyl 41604-19-7 Lab Scale Flurbiprofen
54. 1-methyl-1H-indazole-3-carboxylic acid 50890-83-0 Lab Scale Granisetron
55. Endo-9-methyl-9-azabicyclo[3.3.1]nonan-3-amine 76272-56-5 Lab Scale Granisetron
56. Methyl 4-(bromomethyl) benzoate 2417-72-3 Commercial Imatinib
57. 4-(4-methyl piperazinomethyl) benzoicacid dihydrochloride 106261-49-8 Commercial Imatinib
58. N-(5-Amino-2-methylphenyl)-4-(3-pyridyl)-2-pyrimidine amine 152460-10-1 Commercial Imatinib
59. 1,4\'-bipiperidine 4897-50-1 Commercial Irinotecan
60. 2-(chloromethyl)-4-methyl quinazoline 109113-72-6 Commercial Linagliptin
61. 8-bromo-3-methyl-1H-purine-2,6(3H,7H)-dione 93703-24-3 Commercial Linagliptin
62. 8-bromo-7-(but-2-ynyl)-3-methyl-1H-purine-2,6(3H,7H)-dione 666816-98-4 Commercial Linagliptin
63. 8-bromo-7-(but-2-ynyl)-3-methyl-1-((4-methylquinazolin-2-yl)methyl)-1H-purine-2,6(3H,7H)-dione 853029-57-9 Commercial Linagliptin
64. (R)-tert-butyl 3-amino piperidine-1-carboxylate 309956-78-3 Commercial Linagliptin
65. N-(8-benzyl-8-aza-bicyclo [3.2.1]oct-3-yl-exo)-2-methylpropanamide 376348-67-3 Lab Scale Maraviroc
66. Boc-4-Amino-L-phenylalanine 55533-24-9 Lab Scale Melphalane
67. 2-(1H-indol-5-yl)-N-methylethanesulfonamide 98623-50-8 Commercial Naratriptan
68. N-methyl-2-(3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-yl) ethane sulfonamide 121679-20-7 Commercial Naratriptan
69. 4- Methyl cinnamic acid methyl ester 866157-50-8 Commercial Ozagrel
70. 4- Bromomethyl cinnamic acid methyl ester 946-99-6 Commercial Ozagrel
71. 1,4,8,11-Tetraazacyclotetradecane (Cyclam) 295-37-4 Lab scale Plerixafor
72. 1,4-Bis(bromomethyl)benzene 623-24-5 Lab scale Plerixafor
73. 3-isobutylglutaric acid 75143-89-4 Commercial Pregabalin
74. 3-carbamoylmethyl-5-hexanoic acid 181289-15-6 Commercial Pregabalin
75. R-(-)-3-carbamoylmethyl-5-hexanoic acid 181289-33-8 Commercial Pregabalin
76. 2,3-dimethyl-2H-indazol-6-amine 44473-72-0 Lab Scale Pazopanib
77. N-(2-chloropyrimidin-4-yl)-N,2,3-trimethyl-2H-indazol-6-amine 444731-75-3 Lab Scale Pazopanib
78. 5-Amino-2-methyl-benzenesulfonamide 6973-09-7 Lab Scale Pazopanib
79. 4-((1H-1,2,4-triazol-1-yl)methyl) benzeneamine 119192-10-8 Commercial Rizatriptan
80. 1-(4-nitrobenzyl)-1H-1,2,4-triazole Commercial Rizatriptan
81. 2-((2-methoxy phenoxy) methyl)oxirane 2210-74-4 Commercial Ranolazine
82. N-(2,6-dimethylphenyl)-2-(piperazin-1-yl)acetamide 5294-61-1 Commercial Ranolazine
83. (S)-3-(1-(dimethyl amino) ethyl)phenol 139306-10-8 Commercial Rivastigmine
84. 3-(Trifluoromethyl)-5,6,7,8-tetrahydro [1,2,4]triazolo[4,3-A]pyrazine hydrochloride 762240-92-6 Commercial Sitagliptin
85. Boc-(R)-3-Amino-4-(2,4,5-Trifluorophenyl)-butyric acid 486460-00-8 Commercial Sitagliptin
86. Boc-(R)-3-Amino-4-(2,4,5-Trifluorophenyl)-butyric acid 486460-00-8 Commercial Sitagliptin
87. (1S,3S,5S)-3-(Aminocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester 361440-67-7 Lab scale Saxagliptin
88. (1S,3S,5S)-2-azabicyclo [3.1.0]hexane-3-carboxamide hydrochloride 709031-39-0 Lab scale Saxagliptin
89. 2-(bromomethyl)-4-fluorobenzonitrile 421552-12-7 Lab scale Trelagliptin
90. 2-((6-chloro-3-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl)-5-fluorobenzonitrile 865759-24-6 Lab scale Trelagliptin
91. 1-(3-Methyl-1-phenyl-5-pyrazolyl)piperazine 401566-79-8 Lab scale Tenelagliptin
92. 5-Fluoro oxindole 56341-41-4 Lab Scale Sunitinib
93. 2-tert-butyl 4-ethyl 3,5-dimethyl-1H-pyrrole-2,4-dicarboxylate 86770-31-2 Lab Scale Sunitinib
94. ethyl 5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxylate 2199-59-9 Lab Scale Sunitinib
95. N-(2-(diethylamino)ethyl)-5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxamide 356068-86-5 Lab Scale Sunitinib
96. (3R,4R)-1-Benzyl-N,4-dimethylpiperidin-3-amine 477600-70-7 Lab Scale Tofacitinib
97. 4-chloro-7H-pyrrolo[2,3-d]pyrimidine 3680-69-1 Lab Scale Tofacitinib
98. N-((3R,4R)-1-benzyl-4-methylpiperidin-3-yl)-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine 477600-73-0 Lab Scale Tofacitinib
99. 2-Amino-2-cyanoacetamide 6719-21-7 Pilot Scale Temazolamide
100. 5-amino-1H-imidazole-4-carboxamide Monohydrate 360-97-4 Pilot Scale Temazolamide
101. 5-Amino-N1-methyl-1H-imidazole-1,4-dicarboxamide 188612-53-5 Pilot Scale Temazolamide
102. 3-Methyl-4-oxo-3,4-dihydroimidazo[5,1-d][1,2,3,5]tetrazine-8-carbonitrile 287964-59-4 Pilot Scale Temazolamide
103. N-Benzoyl-DL-tyrosil-N\',N\'-dipropylamide 57227-09-5 Lab scale Tiropramide
104. (S)-1-(2-chloroacetyl) pyrrolidine-2-carbonitrile 207557-35-5 Commercial Vildagliptin
105. 1-amino-3-hydroxy adamantane 702-82-9 Commercial Vildagliptin
106. 2-Acetylbenzothiophene 22720-75-8 Commercial Zileuton
107. 1-Bromo-3,5-dimethyl adamantane 941-7-7 Lab Scale Memantine
108. 1-Acetamido-3,5-dimethyladamantane 19982-07-1 Lab Scale Memantine
109. 2-Amino-4’-bromobenzophenone 1140-17-6 Lab Scale Bromfenac
110. 1-(2,3-Dihydro-1,4-benzodioxin-2-ylcarbonyl)piperazine hydrochlorid 70918-74-0 Commercial Doxazosin
111. 4-Fluoro-2-nitrobenzonitrile 80517-21-1 Lab Scale Fine chemical
112. 1,4,7-Trimethyl-1,4,7-Triazacyclononane 96556-05-7 Lab Scale Fine chemical
113. propane-1,2,3-triyl tris(4-phenylbutanoate) 611168-24-2 Lab Scale Fine chemical
114. ethyl 2-(4-acetylphenyl)acetate 1528-42-3 Commercial Fine chemical
115. 5-Hydroxyvanillin 3934-87-0 Lab Scale Fine chemical
116. 4-Biphenylacetic acid 5728-52-9 Lab Scale Fine chemical
117. 6-Aminocoumarine hydrochloride 63989-79-7 Lab Scale Fine chemical
118. 7-Azaindole 271-63-6 Lab Scale Fine chemical
119. 5-Bromo-2,2-dimethyl-1,3-benzodioxole 73790-19-9 Lab Scale Fine chemical
120. 2,6-Bis-(trifluromethyl)benzoic acid 24821-22-5 Lab Scale Fine chemical
121. N-Benzoyl-6-aminopurine 400-49-6 Lab Scale Fine chemical
122. 4-Chloro-5-nitrophthalimide 6015-57-2 Lab Scale Fine chemical
123. 1-(2-Carboxyphenyl)pyrrole 10333-68-3 Lab Scale Fine chemical
124. Cyclopropyl phenyl ketone 3481-02-5 Lab Scale Fine chemical
125. 4-Chloro-2-(methylthio)pyrimidine 49844-90-8 Lab Scale Fine chemical
126. Dimethyl-trans-stilbene-4,4’-dicarboxylate 34541-73-6 Lab Scale Fine chemical
127. 2,5-Dimethyl-1-phenylpyrrole-3-carboxaldehyde 83-18-1 Lab Scale Fine chemical
128. 2,2-Diphenylpropylamine HCl 40691-66-5 Lab Scale Fine chemical
129. 6-Aminocoumarine hydrochloride 63989-79-7 Lab Scale Fine chemical
130. 7-Azaindole 271-63-6 Lab Scale Fine chemical
131. 5-Bromo-2,2-dimethyl-1,3-benzodioxole 73790-19-9 Lab Scale Fine chemical
132. 2,6-Bis-(trifluromethyl)benzoic acid 24821-22-5 Lab Scale Fine chemical
133. N-Benzoyl-6-aminopurine 400-49-6 Lab Scale Fine chemical
134. 4-Chloro-5-nitrophthalimide 6015-57-2 Lab Scale Fine chemical
135. 1-(2-Carboxyphenyl)pyrrole 10333-68-3 Lab Scale Fine chemical
136. 5,7-Dihydroxy-4-methylcoumarin 2107-76-8 Lab Scale Fine chemical
137. ( S )-(+)-Diphenylprolinol 22348-32-9 Lab Scale Fine chemical
138. ( R )-(-)-Diphenylprolinol 112068-01-6 Lab Scale Fine chemical
139. 1,3-Diethyl-5-nitroso-6-aminouracil 89073-60-9 Lab Scale Fine chemical
140. 2,4-Dichloro-6-nitroaniline 2683-43-4 Lab Scale Fine chemical
141. 4,5-Dimethyl-2-nitro aniline 6972-71-0 Lab Scale Fine chemical
142. 3,4-Dihydro-5-hydroxycarbostyril 30389-33-4 Lab Scale Fine chemical
143. 1,5-Naphthyridine-2-carboxylic acid 49850-62-6 Lab Scale Fine chemical
144. N-Ethyl-N-methylcarbamoyl chloride 42252-34-6 Lab Scale Fine chemical
145. 2-Ethyltoluene 611-14-3 Lab Scale Fine chemical
146. 3- Ethyltoluene 620-14-4 Lab Scale Fine chemical
147. 4- Ethyltoluene 622-96-8 Lab Scale Fine chemical
148. 3-Furaldehyde 498-60-2 Lab Scale Fine chemical
149. 3-Methylpyridazine 1120-88-3 Lab Scale Fine chemical
150. 4-Nitroindole 97% 4769-97-5 Lab Scale Fine chemical
151. ( S )-(+)-4-Phenyl-2-oxazolidinone 99395-88-7 Lab Scale Fine chemical
152. 4-Aminophthalic acid 5434-21-9 Pilot Scale Fine chemical
153. tert-butyl 4-(2-hydroxyphenyl)piperazine-1-carboxylate 313657-51-1 Lab Scale Fine chemical
154. 4-Trifluoromethyl nicotinic acid 158063-66-2 Lab Scale Fine chemical
155. trans-Boc-4-amino cyclohexane carboxylic acid 53292-89-0 Pilot Scale Fine chemical
156. 1,3-Bis(hydroxyimino) propan-2-one 41886-31-1 Lab Scale Fine chemical
157. 7-methoxy-3-(trifluoromethyl)quinoxalin-2(1H)-one 445498-40-8 Lab Scale Fine chemical
158. 3-ethyl-7-methoxyquinoxalin-2(1H)-one Lab Scale Fine chemical
159. 3-isopropyl-7-methoxy quinoxalin-2(1H)-one 445498-48-6 Lab Scale Fine chemical
160. 7-methoxy-3-methy lquinoxalin-2(1H)-one 117237-99-7 Lab Scale Fine chemical
161. 3-chloro-7-methoxy quinoxalin-2(1H)-one 1263814-66-9 Lab Scale Fine chemical
162. Isovanilline 621-59-0 Pilot Scale Fine chemical
163. Ethyl- 4,4,4-trifluoro-2-butynoate 79424-03-6 Lab Scale Fine chemical
164. Methylene cyclopropane (In THF) 6142-73-0 Lab Scale Fine chemical
165. 2,3-Dichloro-1-propene 78-88-6 Lab Scale Fine chemical
166. 1-Bromo-2-butyne 3355-28-0 Lab Scale Fine chemical
167. 1-Bromo-2-pentyne 16400-32-1 Lab Scale Fine chemical
168. 5-Bromo-1,2,3,4-tetrahydroquinoline hydrochloride 81237-69-6 Lab Scale Fine chemical
169. Ter-Butyl-3-(bromomethyl)phenyl carbamate 118684-32-5 Lab Scale Fine chemical
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